Terbutaline: Difference between revisions

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==General==
==General==
*Type:  
*Type: [[Beta 2 agonist]]
*Dosage Forms:
*Dosage Forms: 1mg/mL injection
*Common Trade Names:


==Adult Dosing==
==Adult Dosing==
===[[Preterm labor]]===
*0.25mg sq q20-30 min, up to 4 doses PRN contractions
===Asthma/Bronchoconstriction===
*0.25mg sq q20 min, up to 3 doses


==Pediatric Dosing==
==Pediatric Dosing==
===Asthma/Bronchoconstriction===
*0.005-0.01mg/kg to max 0.4mg SQ q15-20 min, up to 3 doses; may repeat in 2-6 hours


==Special Populations==
==Special Populations==
*[[Drug Ratings in Pregnancy|Pregnancy Rating]]:
*[[Drug Ratings in Pregnancy|Pregnancy Rating]]: Category C
*Lactation:
*Lactation: Not recommended
*Renal Dosing
*Renal Dosing: n/a
**Adult
*Hepatic Dosing: n/a
**Pediatric
*Hepatic Dosing
**Adult
**Pediatric


==Contraindications==
==Contraindications==
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==Adverse Reactions==
==Adverse Reactions==
===Serious===
===Serious===
*Black box warning against prolonged use for tocolysis (>48-72 hrs)
*Cardiac arrhythmia


===Common===
===Common===
*Agitation, tremor, hyperglycemia, hypokalemia


==Pharmacology==
==Pharmacology==
*Half-life:  
*Onset: 6-15 minutes
*Metabolism:  
*Half-life: 11-16 hours
*Excretion:  
*Metabolism: Hepatic
*Mechanism of Action:
*Excretion: Urine
*Mechanism of Action: Beta 2 agonist, smooth muscle relaxant
 
 
==Indications by Condition==
''The following table is automatically generated from disease/condition pages across WikEM.''
 
{{#ask:[[Has DrugName::Terbutaline]]
|?Has Indication=Indication
|?Has Dose=Dose
|?Has Context=Context
|?Has Route=Route
|?Has Population=Population
|format=table
|headers=plain
|mainlabel=-
|sort=Has Indication
|limit=50
}}


==See Also==
==See Also==
[[Asthma]], [[Preterm Labor]]


==Sources==
==References==
 
Lexicomp
<references/>
<references/>
[[Category:Drugs]]
[[Category:Pharmacology]]

Latest revision as of 21:55, 20 March 2026

General

Adult Dosing

Preterm labor

  • 0.25mg sq q20-30 min, up to 4 doses PRN contractions

Asthma/Bronchoconstriction

  • 0.25mg sq q20 min, up to 3 doses

Pediatric Dosing

Asthma/Bronchoconstriction

  • 0.005-0.01mg/kg to max 0.4mg SQ q15-20 min, up to 3 doses; may repeat in 2-6 hours

Special Populations

  • Pregnancy Rating: Category C
  • Lactation: Not recommended
  • Renal Dosing: n/a
  • Hepatic Dosing: n/a

Contraindications

  • Allergy to class/drug

Adverse Reactions

Serious

  • Black box warning against prolonged use for tocolysis (>48-72 hrs)
  • Cardiac arrhythmia

Common

  • Agitation, tremor, hyperglycemia, hypokalemia

Pharmacology

  • Onset: 6-15 minutes
  • Half-life: 11-16 hours
  • Metabolism: Hepatic
  • Excretion: Urine
  • Mechanism of Action: Beta 2 agonist, smooth muscle relaxant


Indications by Condition

The following table is automatically generated from disease/condition pages across WikEM.

IndicationDoseContextRoutePopulation
Acute asthma exacerbation0.25 mg SC/IM q20min x3Beta-2 agonist (longer-acting)SC/IMAdult
Preterm labor0.25mg SC q20-30min up to 4 doses PRNTocolyticSCAdult
Priapism0.25-0.5 mg SQ or 5-10 mg POBeta-agonist (adjunct)SQ/POAdult

See Also

Asthma, Preterm Labor

References

Lexicomp